SCHEMBL3988092

SCHEMBL3988092

c1ccc2c(c1)NCC21CCN(C2C3CC4CC(C3)CC2C4)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
USP2 O75604 1/20 0.40
OPRM1 P35372 3/20 0.39
OPRL1 P41146 3/20 0.39
AVPR1A P37288 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KCNH2 Q12809 1/20 0.36
HDAC1 Q13547 1/20 0.36
HSD11B1 P28845 4/20 0.36
KDM1A O60341 1/20 0.35
CYP2A13 Q16696 1/20 0.35
HSD11B2 P80365 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
CCR5 P51681 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PRNP P04156 1/20 0.32
SLC18A3 Q16572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12084354 0.82 KDM4E (0.43) TNKSTNKS2OPRM1OPRL1AVPR1A
SCHEMBL12084848 0.81 OPRM1 (0.42) TNKSTNKS2OPRM1OPRL1AVPR1A
SCHEMBL12084329 0.81 TNKS (0.38) TNKSTNKS2OPRM1OPRL1AVPR1A
SCHEMBL4115045 0.79 HSD11B1 (0.41) USP2OPRM1OPRL1ALDH1A1SMN1; SMN2
SCHEMBL13644096 0.77 TNKS (0.44) TNKSTNKS2OPRM1OPRL1AVPR1A
SCHEMBL30441215 0.77 TNKS (0.43) TNKSTNKS2OPRM1OPRL1AVPR1A
SCHEMBL1222308 0.76 HSD11B1 (0.66) HSD11B1HSD11B2
SCHEMBL1223289 0.76 HSD11B1 (0.55) TNKSTNKS2AVPR1AKCNH2HDAC1
SCHEMBL12084593 0.75 TNKS (0.44) TNKSTNKS2OPRM1OPRL1AVPR1A
SCHEMBL13644048 0.74 TNKS (0.42) TNKSTNKS2OPRM1OPRL1AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2064187-A2 INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 Vitae Pharmaceuticals, Inc. (US) 2009-06-03 EP claimed
WO-2008024497-A2 INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE TYPE 1 VITAE PHARMACEUTICALS, INC. (US) 2008-02-28 WO claimed