SCHEMBL4115045

SCHEMBL4115045

c1ccc2c(c1)CNCC21CCN(C2C3CC4CC(C3)CC2C4)CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.41
USP2 O75604 1/20 0.39
KCNH2 Q12809 1/20 0.38
HDAC1 Q13547 1/20 0.38
SIGMAR1 Q99720 3/20 0.38
SLC18A3 Q16572 3/20 0.37
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
OPRM1 P35372 2/20 0.34
OPRL1 P41146 2/20 0.34
CYP2A13 Q16696 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HSD11B2 P80365 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
OPRK1 P41145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3991405 0.79 SIGMAR1 (0.53) HSD11B1SIGMAR1SLC18A3HTR2AHTR2C
SCHEMBL3988092 0.79 TNKS (0.40) HSD11B1USP2KCNH2HDAC1SIGMAR1
SCHEMBL1222270 0.77 HSD11B1 (0.73) HSD11B1HSD11B2
SCHEMBL1222092 0.77 HSD11B1 (0.53) HSD11B1KCNH2HDAC1HSD11B2
SCHEMBL11939419 0.76 OPRM1 (0.42) KCNH2HDAC1SIGMAR1SLC18A3SMN1; SMN2
SCHEMBL17969883 0.76 KCNH2 (0.43) KCNH2HDAC1SIGMAR1HTR2AHTR2C
SCHEMBL4119925 0.76 KDM4E (0.44) HSD11B1USP2SIGMAR1SLC18A3ALDH1A1
SCHEMBL2256944 0.75 HTR2A (0.43) KCNH2HDAC1HTR2AHTR2CHTR2B
SCHEMBL29526055 0.75 HTR2A (0.43) KCNH2HDAC1HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL30090414 0.74 HTR2A (0.42) KCNH2HDAC1HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2064187-A2 INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 Vitae Pharmaceuticals, Inc. (US) 2009-06-03 EP disclosed
WO-2008024497-A2 INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE TYPE 1 VITAE PHARMACEUTICALS, INC. (US) 2008-02-28 WO disclosed