SCHEMBL3989130

SCHEMBL3989130

O=C=Nc1ccc(CCCl)cc1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.63
TSHR P16473 1/20 0.63
P2RY6 Q15077 1/20 0.47
CYP1A2 P05177 1/20 0.46
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TRPA1 O75762 1/20 0.37
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL733010 0.87 CYP3A4 (0.74) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL1900351 0.83 CYP3A4 (0.68) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL93415 0.83 CYP3A4 (0.68) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL7898757 0.83 CYP3A4 (0.68) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL11061694 0.81 CYP3A4 (0.65) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL11723360 0.81 CYP3A4 (0.65) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL4600058 0.79 CYP3A4 (0.63) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL27930613 0.79 CYP3A4 (0.63) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL93144 0.79 CYP3A4 (0.63) CYP3A4TSHRP2RY6CYP1A2MAPK1
SCHEMBL19943 0.78 CYP3A4 (1.00) CYP3A4TSHRP2RY6CYP1A2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009061131-A2 NOVEL TRICYCLIC DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME JE IL PHARMACEUTICAL CO., LTD. (KR) 2009-05-14 WO disclosed