SCHEMBL3994601

SCHEMBL3994601

CC(C)c1ccc(-c2ccc(C=O)nc2-c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.44
PDE10A Q9Y233 1/20 0.44
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
ERN1 O75460 1/20 0.40
TYR P14679 1/20 0.39
S1PR3 Q99500 2/20 0.36
MAPT P10636 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
LMNA P02545 2/20 0.35
RAB9A P51151 1/20 0.35
PAX8 Q06710 1/20 0.35
NOD2 Q9HC29 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ERBB2 P04626 1/20 0.35
USP2 O75604 1/20 0.35
PTGS2 P35354 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2830315 0.86 CCR1 (0.42) S1PR3MEN1KMT2ALMNARAB9A
SCHEMBL2835431 0.84 TDP1 (0.49) DHODHS1PR3MAPTMEN1KMT2A
SCHEMBL2830330 0.80 S1PR3 (0.54) S1PR3MAPTLMNARAB9A
SCHEMBL2831010 0.78 S1PR3 (0.53) PDE10AS1PR3MAPTLMNARAB9A
SCHEMBL2832332 0.77 KIF11 (0.47) DHODHMAPK13MAPK12MAPK11MAPK14
SCHEMBL3997120 0.75 S1PR3 (0.44) DHODHPDE10AMAPK13MAPK12MAPK11
SCHEMBL9876332 0.74 PTGS2 (0.47) MAPK13MAPK12MAPK11MAPK14MAPT
SCHEMBL2836985 0.73 GABRA1 (0.44) DHODHPDE10AMAPK13MAPK12MAPK11
SCHEMBL5365268 0.73 MAPT (0.51) MAPTMEN1KMT2ALMNARAB9A
SCHEMBL27320637 0.72 PSMB5 (0.42) ERN1MEN1KMT2ARAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066633-A1 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST AND/OR ANTAGONIST BIOLOGICAL ACTIVITY Allergan, Inc. (US) 2009-06-10 EP disclosed
WO-2008030843-A1 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST AND/OR ANTAGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2008-03-13 WO disclosed