SCHEMBL3997682

SCHEMBL3997682

NC(=S)N(CCCN1CCCCC1)NC(=O)c1cn(-c2ccccc2)c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.45
HDAC2 Q92769 3/20 0.45
NR4A2 P43354 1/20 0.42
HTR3A P46098 1/20 0.41
HTR7 P34969 8/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
GFER P55789 1/20 0.39
RAD52 P43351 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CNR1 P21554 2/20 0.38
CNR2 P34972 2/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3997685 0.78 HDAC1 (0.50) HDAC1HDAC2NR4A2HTR3AKDM4E
SCHEMBL4131795 0.74 ALDH1A1 (0.50) ALDH1A1
SCHEMBL3996474 0.70 NR4A2 (0.64) HDAC1HDAC2NR4A2HTR3AHTR7
SCHEMBL4241227 0.68 SIGMAR1 (0.45) KDM4EALDH1A1SMN1; SMN2GAA
SCHEMBL27806604 0.68 PARP1 (0.53) HDAC1HDAC2NR4A2HTR7GAA
SCHEMBL579555 0.66 NR4A2 (0.65) HDAC1HDAC2NR4A2HTR3AHTR7
SCHEMBL4003298 0.66 CHEK2 (0.48) HDAC1
SCHEMBL27381209 0.66 LIPG (0.53) HDAC1HDAC2NR4A2HTR3AHTR7
SCHEMBL10321788 0.66 NR4A2 (0.64) HDAC1HDAC2NR4A2HTR3AKDM4E
SCHEMBL407789 0.66 HDAC1 (0.65) HDAC1HDAC2NR4A2HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071577-A1 OXADIAZOLE DERIVATIVES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS GLAXO GROUP LIMITED (GB) 2009-06-11 WO disclosed