SCHEMBL3999574

SCHEMBL3999574

FC(F)(F)c1cccc(-c2cccc(Cl)n2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.60
KDM1A O60341 2/20 0.55
IDO1 P14902 1/20 0.51
KMO O15229 2/20 0.51
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
XDH P47989 1/20 0.49
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
HPGD P15428 2/20 0.48
HSD17B10 Q99714 2/20 0.48
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
THRB P10828 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
TSHR P16473 1/20 0.48
STAT6 P42226 1/20 0.48
HTT P42858 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16538337 0.82 SCN9A (0.46)
SCHEMBL4787 0.79 CTSS (0.60) CTSSKDM1AIDO1KMOKDM4E
SCHEMBL2615262 0.79 CTSS (0.60) CTSSKDM1AIDO1KMOKDM4E
SCHEMBL6256565 0.79 CTSS (0.60) CTSSKDM1AIDO1KMOKDM4E
SCHEMBL3970891 0.78 CNR2 (0.53) CTSSKDM1AIDO1KMOKDM4E
SCHEMBL13854087 0.77 CTSS (0.58) CTSSKDM1AIDO1KMOKDM4E
SCHEMBL9971080 0.77 CTSS (0.57) CTSSKDM1AIDO1KMOKDM4E
SCHEMBL601224 0.77 KMO (0.61) CTSSKDM1AIDO1KMOKDM4E
SCHEMBL38663516 0.76 CNR2 (0.50) IDO1KMOKDM4EALDH1A1CNR2
SCHEMBL9954071 0.76 CTSS (1.00) CTSSKDM1AIDO1KMOKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009068652-A1 2, 6-DISUBSTITUTED PYRIDINES AND 2, 4-DISUBSTITUTED PYRIMIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed
WO-2009068652-A1 2, 6-DISUBSTITUTED PYRIDINES AND 2, 4-DISUBSTITUTED PYRIMIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed