SCHEMBL6256565

SCHEMBL6256565

Nc1cccc(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.60
ASIC3 Q9UHC3 1/20 0.56
XDH P47989 1/20 0.56
KDM1A O60341 3/20 0.52
IDO1 P14902 1/20 0.51
KMO O15229 2/20 0.51
ADORA2A P29274 2/20 0.50
ADORA1 P30542 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
TLR8 Q9NR97 1/20 0.48
PIK3CD O00329 1/20 0.47
PIK3CA P42336 1/20 0.47
PIK3CG P48736 1/20 0.47
IKBKB O14920 1/20 0.47
BRD4 O60885 1/20 0.47
ATR Q13535 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1800349 0.82 ASIC3 (0.60) ASIC3ADORA2A
SCHEMBL18039077 0.82 ASIC3 (0.47) CTSSASIC3XDHKDM1AIDO1
SCHEMBL1358158 0.80 XDH (0.57) CTSSXDHKDM1AIDO1KMO
SCHEMBL2615262 0.79 CTSS (0.60) CTSSXDHKDM1AIDO1KMO
SCHEMBL4787 0.79 CTSS (0.60) CTSSXDHKDM1AIDO1KMO
SCHEMBL3999574 0.79 CTSS (0.60) CTSSXDHKDM1AIDO1KMO
SCHEMBL2302878 0.79 CTSS (0.56) CTSSXDHKDM1AIDO1KMO
SCHEMBL2788482 0.79 CCNT1 (0.63) CTSSXDHKDM1AIDO1KMO
SCHEMBL7711733 0.79 ADORA2A (0.53) CTSSXDHKDM1AIDO1ADORA2A
SCHEMBL10853666 0.78 CNR2 (0.53) CTSSXDHKDM1AIDO1KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed