SCHEMBL400222

SCHEMBL400222

c1ccc(COc2ccc(-c3nn[nH]n3)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.67
LMNA P02545 1/20 0.64
ALDH1A1 P00352 2/20 0.63
TP53 P04637 1/20 0.63
XDH P47989 2/20 0.61
GP6 Q9HCN6 2/20 0.61
CYP19A1 P11511 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.55
HPGDS O60760 1/20 0.54
ADH5 P11766 1/20 0.53
HPGD P15428 1/20 0.52
TAS2R14 Q9NYV8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1249156 0.89 KMT2A (0.61) KMT2ALMNAALDH1A1TP53XDH
SCHEMBL1250582 0.85 XDH (0.72) KMT2ALMNAXDH
SCHEMBL1248713 0.84 SLC22A12 (0.68) XDHGP6
SCHEMBL12458012 0.82 GP6 (0.49) KMT2ALMNAGP6HPGDS
SCHEMBL1249112 0.81 KMT2A (0.62) KMT2ALMNAALDH1A1GP6L3MBTL1
SCHEMBL1248177 0.80 GP6 (0.56) KMT2ALMNAALDH1A1TP53GP6
SCHEMBL31530110 0.80 LMNA (0.62) KMT2ALMNAALDH1A1TP53XDH
SCHEMBL7901106 0.79 GRIK1 (0.55) GP6
SCHEMBL1249214 0.79 RHEB (0.51) KMT2ALMNAGP6
SCHEMBL4667928 0.78 LMNA (0.51) KMT2ALMNAXDHCYP2C19L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
CN-101056628-B Ester derivatives and medicinal use thereof JAPAN TOBACCO INC 2011-05-25 CN disclosed
US-7879893-B2 Zinc binding ligand; sustained release of insulin NOVO NORDISK A/S (DK) 2011-02-01 US disclosed
CN-101056628-A Ester derivatives and medicinal use thereof JAPAN TOBACCO INC (JP) 2007-10-17 CN disclosed
EP-1803452-A1 ESTER DERIVATIVE AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2007-07-04 EP disclosed
US-20060089392-A1 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2006-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089392-A1 Ester derivatives and medicinal use thereof MTTP, CETP, LIPA KMT2A 3181/4885LMNA 2858/4885ALDH1A1 421/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.