SCHEMBL4005894

SCHEMBL4005894

NCc1ccccc1-c1c[c]c2ccccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.41
LOXL2 Q9Y4K0 1/20 0.38
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
ATR Q13535 2/20 0.34
UBE2T Q9NPD8 1/20 0.33
ASIC3 Q9UHC3 1/20 0.33
PNMT P11086 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GLA P06280 2/20 0.32
HPGD P15428 2/20 0.32
CASP1 P29466 2/20 0.32
CASP7 P55210 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HSD17B10 Q99714 2/20 0.32
CHRM2 P08172 1/20 0.32
ADRA2A P08913 1/20 0.32
ADORA3 P0DMS8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4875167 0.77 MAPT (0.46) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL4010186 0.76 SMN1; SMN2 (0.43) KDM4EALDH1A1SMN1; SMN2HSD17B10RAB9A
SCHEMBL21483573 0.73 NPC1 (0.47) DPP4NOS2KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL28782153 0.72 MEN1 (0.49) DPP4NOS3NOS1NOS2KDM4E
SCHEMBL234452 0.71 ACHE (0.47) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL8087257 0.70 CYP1A2 (0.46) LOXL2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL29133411 0.68 DHODH (0.46) KDM4EALDH1A1HPGDSMN1; SMN2ACHE
SCHEMBL4875157 0.68 RAB9A (0.46) NOS2KDM4EALDH1A1GLAHPGD
SCHEMBL8090146 0.68 ALDH1A1 (0.38) KDM4EALDH1A1GLAHPGDCASP1
SCHEMBL8102371 0.67 KDM4E (0.50) KDM4EALDH1A1HPGDSMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009082346-A1 NEW ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS AND USES IN TREATMENTS OF OBESITY AND DIABETES MELLITUS - 087 ASTRAZENECA AB (SE) 2009-07-02 WO claimed
WO-2009082346-A1 NEW ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS AND USES IN TREATMENTS OF OBESITY AND DIABETES MELLITUS - 087 ASTRAZENECA AB (SE) 2009-07-02 WO disclosed