SCHEMBL4007809

SCHEMBL4007809

COC(=O)C(=CC1CC1)C(=O)OC

nearest known ligand 0.80

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.35
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
APP P05067 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15913328 0.91 GRIK1 (0.33) RECQLALDH1A1
SCHEMBL15913809 0.89 NPSR1 (0.36) RECQLMAPT
SCHEMBL10471560 0.80 NPSR1 (0.33) RECQLALDH1A1
SCHEMBL10471561 0.80 NPSR1 (0.33) RECQLALDH1A1
SCHEMBL7623965 0.77 ALDH1A1 (0.31) ALDH1A1
SCHEMBL9421764 0.77 ALDH1A1 (0.31) ALDH1A1
SCHEMBL27713674 0.77 ALDH1A1 (0.31) ALDH1A1
SCHEMBL4769947 0.77 CES2 (0.39)
SCHEMBL4014089 0.77 GRIK1 (0.32) ALDH1A1MAPT
SCHEMBL4769941 0.77 CES2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080248-A1 SUBSTITUTED 2-PHENYLPYRIMIDINE-5-CARBOXYLIC ACIDS AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed
EP-0847974-B1 Process for the preparation of cyclopropylacetylene and its derivatives KURARAY CO (JP) 2002-06-05 EP disclosed
US-5955627-A Process for the preparation of cyclopropylacetylene derivatives KURARAY CO., LTD. (JP) 1999-09-21 US disclosed
EP-0847974-A1 Process for the preparation of cyclopropylacetylene and its derivatives KURARAY CO., LTD. (JP) 1998-06-17 EP disclosed