SCHEMBL4010282

SCHEMBL4010282

CCCC1N=C(CC)C(c2ccc(OC(C)C)cc2)=CN1Cc1ccc(-c2ccccc2-c2noc(=O)[nH]2)cc1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARG P37231 8/20 0.43
AGTR1 P30556 2/20 0.43
KCNH2 Q12809 1/20 0.41
LTB4R2 Q9NPC1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016474 0.92 PPARG (0.45) PPARGAGTR1KCNH2LTB4R2
SCHEMBL4016392 0.88 PPARG (0.47) PPARGKCNH2LTB4R2
SCHEMBL4011200 0.84 LTB4R2 (0.42) PPARGLTB4R2
SCHEMBL4016049 0.81 PPARG (0.43) PPARGAGTR1KCNH2LTB4R2
SCHEMBL4017111 0.78 AGTR1 (0.40) PPARGAGTR1
SCHEMBL4010608 0.76 AGTR1 (0.45) PPARGAGTR1
SCHEMBL4016033 0.76 AGTR1 (0.49) PPARGAGTR1KCNH2LTB4R2
SCHEMBL4008051 0.76 SLC33A1 (0.47) AGTR1
SCHEMBL4016610 0.74 SLC33A1 (0.46) AGTR1
SCHEMBL4016519 0.74 SLC33A1 (0.47) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed