SCHEMBL4016392

SCHEMBL4016392

CCCCC1N=C(C)C(c2ccc(OC(C)C)cc2)=CN1Cc1ccc(-c2ccccc2-c2noc(=O)[nH]2)cc1

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 14/20 0.47
KCNH2 Q12809 1/20 0.45
LTB4R2 Q9NPC1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016474 0.95 PPARG (0.45) PPARGKCNH2LTB4R2
SCHEMBL4010282 0.88 PPARG (0.43) PPARGKCNH2LTB4R2
SCHEMBL4016049 0.86 PPARG (0.43) PPARGKCNH2LTB4R2
SCHEMBL4158457 0.83 LTB4R2 (0.45) PPARGLTB4R2
SCHEMBL4014474 0.81 LTB4R2 (0.49) PPARGKCNH2LTB4R2
SCHEMBL1896460 0.75 PPARG (0.70) PPARGKCNH2
SCHEMBL4016389 0.75 PPARG (0.58) PPARGKCNH2
SCHEMBL1893693 0.74 PPARG (0.70) PPARGKCNH2
SCHEMBL4008051 0.73 SLC33A1 (0.47)
SCHEMBL1890861 0.73 PPARG (0.64) PPARGKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed