SCHEMBL401081

SCHEMBL401081

c1ccc2[nH]c(Cc3cc4ccccc4[nH]3)cc2c1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.69
AHR P35869 2/20 0.62
HRH3 Q9Y5N1 1/20 0.58
MTNR1A P48039 1/20 0.54
MTNR1B P49286 1/20 0.54
PCSK9 Q8NBP7 5/20 0.53
AOC3 Q16853 1/20 0.52
HRH4 Q9H3N8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29403791 1.00 LOXL2 (0.69) LOXL2AHRHRH3MTNR1AMTNR1B
SCHEMBL28338445 1.00 LOXL2 (0.69) LOXL2AHRHRH3MTNR1AMTNR1B
SCHEMBL28335219 0.98 LOXL2 (0.67) LOXL2AHRHRH3MTNR1AMTNR1B
SCHEMBL7169246 0.91 LOXL2 (0.69) LOXL2AHRHRH3MTNR1AMTNR1B
SCHEMBL31059889 0.91 LOXL2 (0.69) LOXL2AHRHRH3MTNR1AMTNR1B
SCHEMBL30105384 0.87 LOXL2 (0.60) LOXL2AHRPCSK9
SCHEMBL3193871 0.87 LOXL2 (0.60) LOXL2AHRPCSK9
SCHEMBL17508513 0.87 AHR (0.55) LOXL2AHRHRH3MTNR1AMTNR1B
SCHEMBL6860219 0.86 LOXL2 (0.64) LOXL2AHRHRH3MTNR1AMTNR1B
Bromide SCHEMBL30437340 0.86 LOXL2 (0.58) LOXL2AHRPCSK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2090 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137715-A1 AQUEOUS FORMULATION INCLUDING DISSOLVED HYDROGEN GAS AND MINERALS AND ADDITIVES BEST PLANET SCIENCE LLC (US) 2026-05-21 US claimed
EP-4363043-B1 COMPOSITIONS FOR USE IN METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-04-22 EP claimed
US-12594421-B2 Compositions and methods for increasing cancer cell sensitivity to alternating electric fields NOVOCURE GMBH (CH) 2026-04-07 US claimed
EP-4694699-A2 COMPOSITIONS AND METHODS OF CONTROLLING MAMMALIAN SATIETY VitaKey Inc. (US) 2026-02-18 EP claimed
US-12527765-B2 Composition comprising a diindolylmethane and a retinoid to treat a skin condition SKINTECH LIFE SCIENCE LIMITED (GB) 2026-01-20 US claimed
US-12527804-B2 Microemulsion delivery systems for alcohol-soluble species including DHEA, pregnenolone, and chrysin for reducing menopausal symptoms Quicksilver Scientific, Inc. (US) 2026-01-20 US claimed
EP-4676470-A2 DILEUCINE COMPOSITIONS AND METHODS OF USE THEREOF Ingenious Ingredients, LP (US) 2026-01-14 EP claimed
US-20250339680-A1 COMPOSITIONS AND METHODS FOR INCREASING CANCER CELL SENSITIVITY TO ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2025-11-06 US claimed
WO-2025151636-A2 SPRINKLE PREPARATIONS VITAKEY INC. (US) 2025-07-17 WO claimed
WO-2025133964-A1 A NUTRACEUTICAL FORMULATION TO TREAT HORMONAL IMBALANCES AND MENSTRUAL DISORDERS PATODIA RAMESH (IN) 2025-06-26 WO claimed
WO-2003034992-A2 DIINDOLYLMETHANE FOR THE TREATMENT OF HPV INFECTION BIORESPONSE, L.L.C. (US) 2003-05-01 WO claimed
US-6544564-B1 Cytotoxic pharmaceutical composition FARLEY MICHAEL DONALD (US) 2003-04-08 US claimed
WO-2002080906-A1 PREVENTION AND TREATMENT OF ENDOMETRIOSIS WITH ARYL HYDROCARBON RECEPTOR BINDING LIGANDS CEDARS-SINAI MEDICAL CENTER (US) 2002-10-17 WO claimed
US-20020147155-A1 Prevention and treatment of endometriosis with aryl hydrocarbon receptor binding ligands CEDARS-SINAI MEDICAL CENTER 2002-10-10 US claimed
US-6399645-B1 Chemoprevention and treatment of cervical or vaginal neoplasia BELL MARIA (US) 2002-06-04 US claimed
US-20020058648-A1 Estrogenic substances combined with cruciferous indole compounds HAMMERLY MILTON (US) 2002-05-16 US claimed
WO-2002028832-A2 DIINDOLYLMETHANE AND C-SUBSTITUTED DIINDOLYLMETHANE COMPOSITIONS AND METHODS FOR THE TREATMENT OF MULTIPLE CANCERS THE TEXAS A & M UNIVERSITY SYSTEM (US) 2002-04-11 WO claimed
EP-1067913-A1 COMPOSITIONS AND METHODS OF ADJUSTING STEROID HORMONE METABOLISM THROUGH FACILITATED ABSORPTION OF HYDROPHOBIC DIETARY COMPOUNDS Bioresponse, L.L.C. (US) 2001-01-17 EP claimed
US-6086915-A HEATING THE SOLUBILIZING EMULSIFIER, ADDING SOLVENT AND ONE OR MORE PHOSPHOLIPID SURFACTANTS, DISSOLVING IN THIS SOLUTION ONE OR MORE HYDROPHOBIC PHYTOCHEMICALS, ADDING ENCAPSULATORS, FORMING MICROEMULSION, SPRAY DRYING THE SOLUTION BIORESPONSE L.L.C. (US) 2000-07-11 US claimed
WO-1999049851-A1 COMPOSITIONS AND METHODS OF ADJUSTING STEROID HORMONE METABOLISM THROUGH FACILITATED ABSORPTION OF HYDROPHOBIC DIETARY COMPOUNDS BIORESPONSE, L.L.C. (US) 1999-10-07 WO claimed