SCHEMBL4012143

SCHEMBL4012143

Cc1cc(-c2cc(O)ccc2Cl)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.40
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
NR4A2 P43354 1/20 0.39
PDE2A O00408 1/20 0.39
PDE10A Q9Y233 1/20 0.39
RORC P51449 3/20 0.38
ACVR1 Q04771 1/20 0.38
CRHR1 P34998 2/20 0.38
CD38 P28907 2/20 0.38
CYP3A4 P08684 1/20 0.38
TRPV1 Q8NER1 4/20 0.37
BDKRB2 P30411 2/20 0.37
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012780 0.86 CD38 (0.41) ESR1GAAMAPTACVR1CD38
SCHEMBL4017818 0.85 NR4A2 (0.54) GAAMAPTNR4A2PDE2APDE10A
SCHEMBL4012142 0.83 ENPP1 (0.44) GAAMAPTNR4A2PDE2APDE10A
SCHEMBL2451399 0.81 ESR1 (0.42) ESR1PDE2APDE10ACRHR1TRPV1
SCHEMBL4009254 0.81 NR1H2 (0.47) ESR1MAPTCYP3A4
SCHEMBL4014169 0.81 PIK3CD (0.46) ESR1GAAMAPTCD38CYP3A4
SCHEMBL4010841 0.78 RORC (0.40) ESR1RORCBDKRB2
SCHEMBL19610603 0.78 MAPT (0.57) ESR1MAPTNR4A2RORCCRHR1
SCHEMBL4019153 0.77 NR4A2 (0.50) GAAMAPTNR4A2CRHR1CD38
SCHEMBL4010226 0.77 NR1H2 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed