SCHEMBL4010898

SCHEMBL4010898

O=S(=O)(Oc1c(F)c(F)c(F)c(F)c1F)c1cccc(CBr)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HTR6 P50406 2/20 0.33
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
CYP19A1 P11511 1/20 0.32
NPC1 O15118 1/20 0.32
TNF P01375 1/20 0.32
RAB9A P51151 1/20 0.32
NOD1 Q9Y239 1/20 0.32
F2 P00734 1/20 0.32
TRPA1 O75762 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
TAS2R14 Q9NYV8 1/20 0.30
CYP4F2 P78329 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27765107 0.88 HTR6 (0.37) CA1CA2CA9MEN1KMT2A
SCHEMBL4565530 0.80 KAT6A (0.39) CA1CA2CA9MEN1KMT2A
SCHEMBL31039994 0.79 HTR6 (0.44) CA1CA2CA9MEN1KMT2A
SCHEMBL4016980 0.76 F2 (0.44) CA1CA2CA9MEN1KMT2A
SCHEMBL4119819 0.75 TDP1 (0.48) CA1CA2CA9KMT2AL3MBTL1
SCHEMBL22829013 0.74 CA1 (0.38) CA1CA2CA9HTR6SCN5A
SCHEMBL27765108 0.74 CA2 (0.33) CA1CA2CA9HTR6SCN5A
SCHEMBL11207039 0.73 NPC1 (0.42) CA1CA2MEN1KMT2AL3MBTL1
SCHEMBL31708776 0.73 NPC1 (0.42) CA1CA2MEN1KMT2AL3MBTL1
SCHEMBL28060767 0.73 HTR6 (0.55) CA1CA2MEN1KMT2AHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed