SCHEMBL4013074

SCHEMBL4013074

CCS(=O)(=O)c1cc(F)cc(Oc2ccc(F)c(-c3ccnc4c(OC)cccc34)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 7/20 0.42
NR1H3 Q13133 7/20 0.42
RXRA P19793 1/20 0.40
SCN9A Q15858 4/20 0.39
AXL P30530 1/20 0.38
MAPK14 Q16539 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
FLT1 P17948 1/20 0.37
FLT4 P35916 1/20 0.37
KDR P35968 1/20 0.37
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.36
HTT P42858 2/20 0.36
RAB9A P51151 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017304 0.92 NR1H2 (0.46) NR1H2NR1H3RXRASCN9AAXL
SCHEMBL4014203 0.91 NR1H2 (0.44) NR1H2NR1H3RXRASCN9AAXL
SCHEMBL4011231 0.91 NR1H2 (0.47) NR1H2NR1H3RXRASCN9AAXL
SCHEMBL4012502 0.88 NR1H2 (0.53) NR1H2NR1H3RXRASCN9APTGDR2
SCHEMBL4012903 0.87 NR1H2 (0.44) NR1H2NR1H3RXRAPTGDR2
SCHEMBL4010852 0.84 NR1H2 (0.56) NR1H2NR1H3RXRAAXLMAPK14
SCHEMBL4015147 0.83 NR1H2 (0.50) NR1H2NR1H3RXRAAXLMAPK14
SCHEMBL4013490 0.82 NR1H2 (0.52) NR1H2NR1H3RXRASCN9AAXL
SCHEMBL4011122 0.81 NR1H2 (0.58) NR1H2NR1H3RXRASCN9AAXL
SCHEMBL4010720 0.80 NR1H2 (0.52) NR1H2NR1H3RXRAPTGDR2FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed