SCHEMBL4013276

SCHEMBL4013276

Clc1cccc2c(-c3cccc(Br)c3)ccnc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.53
NR1H3 Q13133 3/20 0.53
NR4A2 P43354 1/20 0.49
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
NUDT1 P36639 4/20 0.40
PIK3CD O00329 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPK14 Q16539 2/20 0.39
GCGR P47871 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
CCR1 P32246 1/20 0.38
CCR8 P51685 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DYRK1A Q13627 1/20 0.38
HTT P42858 2/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP3A4 P08684 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3357542 0.85 IDO1 (0.42) NR1H2NR1H3IDO1TDO2NUDT1
SCHEMBL28021043 0.82 NR4A2 (0.56) NR1H2NR1H3NR4A2SMN1; SMN2KDM4E
SCHEMBL4016535 0.82 PIK3CD (0.61) NR1H2NR1H3NR4A2NUDT1PIK3CD
SCHEMBL16675083 0.81 IDO1 (0.43) NR1H2NR1H3IDO1TDO2PIK3CD
SCHEMBL25740852 0.79 CYP2A6 (0.50) NR4A2IDO1SMN1; SMN2MAPK14GCGR
SCHEMBL4012984 0.78 NR1H2 (0.62) NR1H2NR1H3IDO1TDO2PIK3CD
SCHEMBL27809134 0.75 NR4A2 (0.51) NR1H2NR1H3NR4A2PIK3CDSMN1; SMN2
SCHEMBL4012775 0.74 NR1H2 (0.77) NR1H2NR1H3NR4A2CYP2C9
SCHEMBL18695357 0.74 CCR1 (0.50) IDO1TDO2PIK3CDSMN1; SMN2KDM4E
SCHEMBL4014159 0.73 NR4A2 (0.61) NR1H2NR1H3NR4A2SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed