SCHEMBL4016535

SCHEMBL4016535

Oc1cccc(-c2ccnc3c(Cl)cccc23)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.61
NR1H2 P55055 1/20 0.53
NR1H3 Q13133 1/20 0.53
NR4A2 P43354 1/20 0.49
CDC7 O00311 1/20 0.47
HSD17B1 P14061 4/20 0.46
HSD17B2 P37059 4/20 0.46
MMP14 P50281 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
TP53 P04637 2/20 0.44
HSP90AA1 P07900 2/20 0.44
CYP3A4 P08684 2/20 0.44
MAPT P10636 2/20 0.44
ALOX15 P16050 2/20 0.44
ALOX12 P18054 2/20 0.44
SLC6A2 P23975 2/20 0.44
OPRK1 P41145 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27809134 0.84 NR4A2 (0.51) PIK3CDNR1H2NR1H3NR4A2MMP14
SCHEMBL28021043 0.82 NR4A2 (0.56) NR1H2NR1H3NR4A2KDM4EALDH1A1
SCHEMBL4011409 0.82 PIK3CD (0.61) PIK3CDNR1H2NR1H3CDC7HSD17B1
SCHEMBL4011946 0.82 NR4A2 (0.49) PIK3CDNR1H2NR1H3NR4A2MMP14
SCHEMBL4013276 0.82 NR1H2 (0.53) PIK3CDNR1H2NR1H3NR4A2MMP14
SCHEMBL4013369 0.82 PIK3CD (0.65) PIK3CDNR1H2NR1H3CDC7HSD17B1
SCHEMBL6558762 0.81 PIK3CD (0.60) PIK3CDCDC7HSD17B1HSD17B2CYP3A4
SCHEMBL4037106 0.79 PIK3CD (0.66) PIK3CDCDC7MMP14KDM4EMEN1
SCHEMBL4013567 0.78 PIK3CD (0.57) PIK3CDCDC7HSD17B1HSD17B2HTR1A
SCHEMBL4016601 0.78 PIK3CD (0.57) PIK3CDNR1H2NR1H3CDC7HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed