SCHEMBL4013295

SCHEMBL4013295

COc1ccc(-c2cnc(N)c(-c3nc4ccccc4[nH]3)n2)cc1S(=O)(=O)N1CCCC1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATR Q13535 19/20 0.57
PRKDC P78527 1/20 0.57
ATM Q13315 1/20 0.57
CLK1 P49759 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4452119 0.93 ATR (0.61) ATRPRKDCATM
SCHEMBL2483748 0.83 ATR (0.71) ATRPRKDCATM
SCHEMBL4008289 0.83 ATR (0.73) ATRPRKDCATM
SCHEMBL4015034 0.82 ATR (0.72) ATRPRKDCATM
SCHEMBL4006573 0.80 ATR (0.59) ATRPRKDCATM
SCHEMBL4003381 0.78 ATR (0.67) ATRPRKDCATM
SCHEMBL13956736 0.76 EGFR (0.53) ATRPRKDCATM
SCHEMBL4297778 0.75 ATR (0.58) ATRPRKDCATM
SCHEMBL4009204 0.74 ATR (0.67) ATRPRKDCATM
SCHEMBL4041720 0.74 ATR (0.82) ATRPRKDCATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO claimed
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO disclosed