SCHEMBL4013423

SCHEMBL4013423

CCS(=O)(=O)c1cc(Br)ccc1C

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 6/20 0.44
EDNRA P25101 6/20 0.44
KMT2A Q03164 1/20 0.44
TSHR P16473 2/20 0.42
GLA P06280 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
PLCG1 P19174 1/20 0.38
LMNA P02545 3/20 0.37
GAA P10253 1/20 0.37
DDR1 Q08345 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14478110 0.84 CA1 (0.51) EDNRBEDNRATSHRGLASMN1; SMN2
SCHEMBL11334245 0.82 ALDH1A1 (0.49) EDNRBEDNRAKMT2ATSHRGLA
SCHEMBL9196907 0.79 EDNRB (0.46) EDNRBEDNRAKMT2ATSHRGLA
SCHEMBL19416657 0.79 HTT (0.46) EDNRBEDNRAKMT2ATSHRSMN1; SMN2
SCHEMBL265203 0.79 EDNRB (0.46) EDNRBEDNRAKMT2ATSHRGLA
SCHEMBL29411241 0.78 TSHR (0.41) EDNRBEDNRAKMT2ATSHRGLA
SCHEMBL264948 0.78 EDNRB (0.45) EDNRBEDNRAKMT2ATSHRGLA
SCHEMBL6465 0.78 EDNRB (0.45) EDNRBEDNRAKMT2ATSHRGLA
SCHEMBL1346608 0.78 CA2 (0.49) EDNRBEDNRAKMT2AALDH1A1CA1
Hydrochloric Acid SCHEMBL28847054 0.76 EDNRB (0.44) EDNRBEDNRAKMT2ATSHRGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed