SCHEMBL264948

SCHEMBL264948

Cc1ccc(Br)cc1S(=O)(=O)Cl

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 4/20 0.45
EDNRA P25101 4/20 0.45
KMT2A Q03164 1/20 0.45
GLA P06280 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
IDH1 O75874 3/20 0.38
LMNA P02545 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
TSHR P16473 1/20 0.37
GAA P10253 1/20 0.36
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
ALDH1A1 P00352 1/20 0.36
S100A4 P26447 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL310277 0.83 CA1 (0.49) EDNRBEDNRAKMT2AGLASMN1; SMN2
SCHEMBL30200885 0.83 CA1 (0.49) EDNRBEDNRAKMT2AGLASMN1; SMN2
SCHEMBL4616375 0.82 LMNA (0.45) KMT2ASMN1; SMN2IDH1LMNACA2
SCHEMBL265203 0.81 EDNRB (0.46) EDNRBEDNRAKMT2AGLASMN1; SMN2
SCHEMBL9196907 0.81 EDNRB (0.46) EDNRBEDNRAKMT2AGLASMN1; SMN2
SCHEMBL6465 0.79 EDNRB (0.45) EDNRBEDNRAKMT2AGLASMN1; SMN2
SCHEMBL1346608 0.79 CA2 (0.49) EDNRBEDNRAKMT2ALMNACA1
SCHEMBL742725 0.78 KMT2A (0.49) EDNRBEDNRAKMT2ASMN1; SMN2LMNA
SCHEMBL197054 0.78 S100A4 (0.48) GLASMN1; SMN2LMNACA1CA2
SCHEMBL198775 0.78 LMNA (0.44) EDNRBEDNRAKMT2AGLASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 178 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025229046-A1 SUBSTITUTED HYDROQUINOLINES FOR THE TREATMENT OF GLIOBLASTOMA MULTIFORME MOLIUS SAGLIK TEKNOLOJILERI ANONIM SIRKETI (TR) 2025-11-06 WO disclosed
EP-4644375-A1 SUBSTITUTED HYDROQUINOLINES FOR THE TREATMENT OF GLIOBLASTOMA MULTIFORME Molius Saglik Teknolojileri Anonim Sirketi (TR) 2025-11-05 EP disclosed
EP-4580621-A2 T-TYPE VOLTAGE-GATED CALCIUM CHANNEL POTENTIATORS The Broad Institute, Inc. (US) 2025-07-09 EP disclosed
WO-2025136671-A1 ANILINO-PYRAZOLE DERIVATIVES, COMPOSITIONS AND METHODS THEREOF ENSEM THERAPEUTICS, INC. (US) 2025-06-26 WO disclosed
CN-120091815-A T-type voltage-gated calcium channel enhancer 广泛研究所股份有限公司 2025-06-03 CN disclosed
EP-4540230-A1 ANILINO-PYRAZOLE DERIVATIVES, COMPOSITIONS AND METHODS THEREOF Ensem Therapeutics, Inc. (US) 2025-04-23 EP disclosed
CN-119384413-A Anilino-pyrazole derivatives, compositions and methods thereof 昂胜医药有限公司 2025-01-28 CN disclosed
US-20240246950-A1 Anilino-Pyrazole Derivatives, Compositions and Methods Thereof Ensem Therapeutics (US) 2024-07-25 US disclosed
US-20240228481-A1 NOVEL SULFONAMIDE SERIES OF QR2 INHIBITORS TO TACKLE OXIDATIVE STRESS AND COGNITIVE DECLINE CARMEL HAIFA UNIVERSITY ECONOMIC CORPORATION LTD. (IL) 2024-07-11 US disclosed
US-11999758-B2 Inhibitors of the YAP/TAZ-TEAD interaction and their use in the treatment of cancer INVENTIVA (FR) 2024-06-04 US disclosed
US-5473067-A Preparation of carbonic anhydrase inhibitors ALCON LABORATORIES, INC. (US) 1995-12-05 US disclosed
US-5424448-A Preparation of carbonic anhydrase inhibitors ALCON LABORATORIES, INC. (US) 1995-06-13 US disclosed
EP-0617038-A1 Preparation of carbonic anhydrase inhibitors ALCON LABORATORIES, INC. (US) 1994-09-28 EP disclosed
US-5344929-A Preparation of carbonic anhydrase inhibitors ALCON LABORATORIES, INC. (US) 1994-09-06 US disclosed
US-4804673-A Fungicidal sulfonyl azoles NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1989-02-14 US disclosed
US-4710509-A IMIDAZOLE AND TRIAZOLE DERIVATIVES; FUNGICIDES NIHON TOKUSHU NOYAKU SEIZO K. K. (JP) 1987-12-01 US disclosed
EP-0237912-A1 Sulfonyl azoles NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1987-09-23 EP disclosed
US-4222937-A Total synthesis of the utero-evacuant substance D,L-zoapatanol ORTHO PHARMACEUTICAL CORP. (US) 1980-09-16 US disclosed
US-4177194-A Total synthesis of the utero-evacuant substance D,L-zoapatanol ORTHO PHARMACEUTICAL CORPORATION (US) 1979-12-04 US disclosed
US-3943157-A Synthesis of codling moth attractant ZOECON CORPORATION (US) 1976-03-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11999758-B2 Inhibitors of the YAP/TAZ-TEAD interaction and their use in the treatment of cancer YAP1, TEAD2, YES1 EDNRB 947/4885EDNRA 1060/4885KMT2A 1435/4885
US-20240228481-A1 NOVEL SULFONAMIDE SERIES OF QR2 INHIBITORS TO TACKLE OXIDATIVE STRESS AND COGNITIVE DECLINE SQOR, NFE2L2, TXNRD2 EDNRB 1636/4885EDNRA 1461/4885KMT2A 354/4885
US-20240246950-A1 Anilino-Pyrazole Derivatives, Compositions and Methods Thereof CDK2, CDK3, CDK4 EDNRB 4042/4885EDNRA 4297/4885KMT2A 1075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.