SCHEMBL4013432

SCHEMBL4013432

CCSc1nc(=O)c(-c2ccccc2)c(C)n1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
MAPK1 P28482 1/20 0.49
PPARG P37231 3/20 0.47
AGTR1 P30556 1/20 0.41
AGTR2 P50052 1/20 0.41
AR P10275 1/20 0.40
ACHE P22303 1/20 0.40
TSHR P16473 1/20 0.40
GRIA2 P42262 1/20 0.39
GRIA4 P48058 1/20 0.39
CNR1 P21554 2/20 0.39
CNR2 P34972 1/20 0.39
PDE3A Q14432 1/20 0.39
DPP4 P27487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1887155 0.87 PPARG (0.48) ALDH1A1PPARGAGTR1AGTR2ACHE
SCHEMBL4012027 0.83 PPARG (0.63) ALDH1A1MAPK1PPARGAGTR1AGTR2
SCHEMBL4010731 0.81 PPARG (0.50) PPARGAGTR1AGTR2ACHECNR1
SCHEMBL13625893 0.80 PPARG (0.48) ALDH1A1PPARGAGTR1AGTR2ACHE
SCHEMBL1889210 0.80 PPARG (0.48) ALDH1A1PPARGAGTR1AGTR2ACHE
SCHEMBL4009715 0.78 PPARG (0.53) PPARGAGTR1AGTR2ACHE
SCHEMBL4017757 0.77 PPARG (0.60) ALDH1A1MAPK1PPARGACHE
SCHEMBL9854355 0.77 PPARG (0.53) ALDH1A1PPARGAGTR1AGTR2
SCHEMBL14208362 0.75 PPARG (0.48) ALDH1A1MAPK1PPARGAGTR1AGTR2
SCHEMBL9264984 0.75 PPARG (0.43) PPARGAGTR1AGTR2ACHEGRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed