Acetic Acid

Acetic Acid

SCHEMBL4013680

CC(=O)O.CC(C)(CCn1cnnc1)NCC(O)c1ccc(OCc2ccccc2)c(CO)c1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 12/20 0.47
ADRB1 P08588 6/20 0.44
ADRB3 P13945 3/20 0.44
CCR5 P51681 1/20 0.39
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014708 0.97 ADRB2 (0.50) ADRB2ADRB1ADRB3CCR5LMNA
SCHEMBL4013682 0.91 ADRB2 (0.40) ADRB2ADRB1ADRB3CCR5LMNA
SCHEMBL4013684 0.88 CCR5 (0.38) ADRB2ADRB1ADRB3CCR5LMNA
SCHEMBL10634796 0.86 ADRB2 (0.47) ADRB2ADRB1CCR5CYP1A2CYP2D6
SCHEMBL11747826 0.85 ADRB2 (0.59) ADRB2ADRB1ADRB3CCR5LMNA
SCHEMBL4014681 0.84 ADRB2 (0.48) ADRB2ADRB1ADRB3CCR5LMNA
SCHEMBL12158787 0.79 ADRB2 (0.58) ADRB2ADRB1CCR5LMNACYP1A2
SCHEMBL4667082 0.79 ADRB2 (0.58) ADRB2ADRB1CCR5LMNACYP1A2
SCHEMBL12158808 0.79 ADRB2 (0.58) ADRB2ADRB1CCR5LMNACYP1A2
SCHEMBL29496355 0.79 ADRB2 (0.58) ADRB2ADRB1CCR5LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7511067-B2 3-hydroxymethyl-4-hydroxy-phenyl-derivatives for the treatment of respiratory diseases BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-31 US disclosed
US-20080132556-A1 3-HYDROXYMETHYL-4HYDROXY-PHENYL- DERIVATIVES FOR THE TREATMENT OF RESPIRATORY DISEASES BOUYSSOU THIERRY 2008-06-05 US disclosed
US-20050234112-A1 3-Hydroxymethyl-4-hydroxy-phenyl-derivatives for the treatment of respiratory diseases BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050234112-A1 3-Hydroxymethyl-4-hydroxy-phenyl-derivatives for the treatment of respiratory diseases PAH, CYP11B1, CYP11B2 ADRB2 117/4885ADRB1 69/4885ADRB3 44/4885
US-20080132556-A1 3-HYDROXYMETHYL-4HYDROXY-PHENYL- DERIVATIVES FOR THE TREATMENT OF RESPIRATORY DISEASES PAH, CYP1A1, CYP11B1 ADRB2 169/4885ADRB1 119/4885ADRB3 110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.