SCHEMBL4014439

SCHEMBL4014439

O=C(OCc1ccncc1)c1ncc[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP17A1 P05093 1/20 0.41
CYP19A1 P11511 1/20 0.41
MAPT P10636 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
POLB P06746 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
NAMPT P43490 1/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28413301 0.88 KMT2A (0.53) KMT2AKDM4ENPC1RAB9APOLB
SCHEMBL432658 0.88 TDP1 (0.53) KMT2ARAB9APOLBTDP1LMNA
SCHEMBL2167257 0.82 POLB (0.50) KMT2AKDM4ENPC1RAB9APOLB
SCHEMBL28415823 0.77 NPC1 (0.42) KMT2ANPC1RAB9APOLBLMNA
SCHEMBL152733 0.75 NUDT1 (0.49) KMT2AKDM4EMAPTNPC1RAB9A
SCHEMBL11181967 0.74 CASP3 (0.58) KMT2AMAPTNPC1RAB9APOLB
SCHEMBL5918034 0.74 RXFP1 (0.61) KMT2AKDM4EMAPTRAB9APOLB
Bromide SCHEMBL29572453 0.73 NUDT1 (0.48) KMT2AKDM4EMAPTNPC1RAB9A
Hydrochloric Acid SCHEMBL29571385 0.73 NUDT1 (0.48) KMT2AKDM4EMAPTNPC1RAB9A
Hydrochloric Acid SCHEMBL6175391 0.73 NUDT1 (0.48) KMT2AKDM4EMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed