SCHEMBL4014540

SCHEMBL4014540

Cc1ccc(O)cc1-c1ccnc2c(C(F)(F)F)cccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 8/20 0.48
NR1H3 Q13133 8/20 0.48
PTGDR2 Q9Y5Y4 1/20 0.45
RXRA P19793 1/20 0.44
ESR1 P03372 2/20 0.44
NCF1 P14598 1/20 0.41
PPARG P37231 1/20 0.40
PIK3CD O00329 1/20 0.39
GSK3A P49840 2/20 0.39
GSK3B P49841 2/20 0.39
DYRK3 O43781 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
CDK1 P06493 1/20 0.39
CDK2 P24941 1/20 0.39
FLT4 P35916 1/20 0.39
CSNK1D P48730 1/20 0.39
CLK2 P49760 1/20 0.39
LIMK1 P53667 1/20 0.39
CSNK2A1 P68400 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4010284 0.87 NR1H2 (0.53) NR1H2NR1H3PTGDR2RXRAESR1
SCHEMBL4009254 0.86 NR1H2 (0.47) NR1H2NR1H3PTGDR2RXRAESR1
SCHEMBL4018678 0.82 NR1H2 (0.47) NR1H2NR1H3PTGDR2RXRANCF1
SCHEMBL1125582 0.81 NR1H2 (0.62) NR1H2NR1H3PTGDR2RXRANCF1
SCHEMBL9033424 0.75 PSMD14 (0.62) NR1H2NR1H3PTGDR2RXRANCF1
SCHEMBL4011829 0.74 NR1H2 (0.66) NR1H2NR1H3RXRA
SCHEMBL1091417 0.74 NCF1 (0.51) NR1H2NR1H3PTGDR2RXRANCF1
SCHEMBL4011442 0.73 NR1H2 (0.58) NR1H2NR1H3RXRA
SCHEMBL4012707 0.72 NR1H2 (0.67) NR1H2NR1H3RXRA
SCHEMBL1124736 0.72 NR1H2 (0.48) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed