SCHEMBL4010284

SCHEMBL4010284

Oc1ccc(F)c(-c2ccnc3c(C(F)(F)F)cccc23)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 8/20 0.53
NR1H3 Q13133 8/20 0.53
PTGDR2 Q9Y5Y4 1/20 0.45
RXRA P19793 1/20 0.44
PIK3CD O00329 1/20 0.42
NCF1 P14598 1/20 0.41
KDM4E B2RXH2 2/20 0.41
PPARG P37231 1/20 0.40
GSK3A P49840 2/20 0.39
GSK3B P49841 2/20 0.39
ESR1 P03372 2/20 0.39
DYRK3 O43781 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
CDK1 P06493 1/20 0.39
CDK2 P24941 1/20 0.39
FLT4 P35916 1/20 0.39
CSNK1D P48730 1/20 0.39
CLK2 P49760 1/20 0.39
LIMK1 P53667 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014540 0.87 NR1H2 (0.48) NR1H2NR1H3PTGDR2RXRAPIK3CD
SCHEMBL4009254 0.86 NR1H2 (0.47) NR1H2NR1H3PTGDR2RXRAPIK3CD
SCHEMBL4012417 0.82 NR1H2 (0.51) NR1H2NR1H3PTGDR2RXRANCF1
SCHEMBL1125582 0.81 NR1H2 (0.62) NR1H2NR1H3PTGDR2RXRAPIK3CD
SCHEMBL2446200 0.81 ESR1 (0.41) NR1H2NR1H3PTGDR2NCF1ESR1
SCHEMBL4013847 0.81 MAPK14 (0.46) PTGDR2PIK3CDKDM4E
SCHEMBL4012780 0.81 CD38 (0.41) NR1H2NR1H3ESR1L3MBTL1
SCHEMBL4299566 0.79 NR1H2 (0.50) NR1H2NR1H3PTGDR2RXRAPIK3CD
SCHEMBL1124663 0.76 NR1H2 (0.55) NR1H2NR1H3PPARGESR1
SCHEMBL16248304 0.75 NCF1 (0.52) NR1H2NR1H3PTGDR2RXRANCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed