SCHEMBL4014474

SCHEMBL4014474

CCCCC1N=C(C)C(C(O)c2ccccc2)=CN1Cc1ccc(-c2ccccc2-c2noc(=O)[nH]2)cc1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 1/20 0.49
PPARG P37231 10/20 0.47
AGTR1 P30556 1/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016392 0.81 PPARG (0.47) LTB4R2PPARGKCNH2
SCHEMBL4158457 0.79 LTB4R2 (0.45) LTB4R2PPARGAGTR1
SCHEMBL4016474 0.77 PPARG (0.45) LTB4R2PPARGAGTR1KCNH2
SCHEMBL1887441 0.73 PPARG (0.69) PPARGAGTR1
SCHEMBL4010717 0.72 PPARG (0.47) LTB4R2PPARG
SCHEMBL4010282 0.71 PPARG (0.43) LTB4R2PPARGAGTR1KCNH2
SCHEMBL4016033 0.70 AGTR1 (0.49) LTB4R2PPARGAGTR1KCNH2
SCHEMBL4302458 0.69 LTB4R2 (0.49) LTB4R2PPARGAGTR1
SCHEMBL4011200 0.69 LTB4R2 (0.42) LTB4R2PPARG
SCHEMBL4011114 0.68 PPARG (0.48) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP claimed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO claimed
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed