SCHEMBL4016963

SCHEMBL4016963

CCCc1nc(CC)c(Oc2cc(F)ccc2F)c(=O)n1Cc1cccc(-c2ccccc2)c1C#N

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 6/20 0.39
AGTR2 P50052 5/20 0.39
PPARG P37231 3/20 0.37
RXRA P19793 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
SQOR Q9Y6N5 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016960 0.87 MAPK14 (0.41) AGTR1AGTR2PPARGKMT2A
SCHEMBL1890287 0.86 PPARG (0.53) AGTR1AGTR2PPARG
SCHEMBL12349180 0.78 AGTR1 (0.45) AGTR1AGTR2
SCHEMBL1895054 0.77 AGTR1 (0.55) AGTR1PPARG
SCHEMBL1891957 0.76 AGTR1 (0.54) AGTR1PPARG
SCHEMBL4016260 0.75 PPARG (0.52) AGTR1PPARG
SCHEMBL4307218 0.73 KDM4E (0.41) PPARGALDH1A1POLBKMT2A
SCHEMBL12349127 0.72 PPARG (0.54) AGTR1AGTR2PPARG
SCHEMBL1895269 0.71 PPARG (0.54) AGTR1PPARG
SCHEMBL1893260 0.71 PPARG (0.51) AGTR1AGTR2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed