SCHEMBL4307218

SCHEMBL4307218

CCCc1nc(C)c(Br)c(=O)n1Cc1cccc(-c2cccc(F)c2)c1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 4/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MAPK14 Q16539 3/20 0.39
CASR P41180 2/20 0.38
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
DPP4 P27487 1/20 0.36
TSHR P16473 1/20 0.36
GFER P55789 1/20 0.36
PPARG P37231 2/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
LMNA P02545 1/20 0.35
GRIA2 P42262 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4015825 0.80 PPARG (0.39) PPARG
SCHEMBL1890409 0.79 PPARG (0.46) ALDH1A1MAPK14POLBKMT2ADPP4
SCHEMBL4011289 0.74 PPARG (0.47) MAPK14DPP4PPARG
SCHEMBL1886369 0.74 PPARG (0.64) PPARG
SCHEMBL1890240 0.74 MAPK14 (0.42) MAPK14DPP4PPARG
SCHEMBL4015830 0.74 POLB (0.42) MAPK14POLBPPARGLMNA
SCHEMBL4016963 0.73 AGTR1 (0.39) ALDH1A1POLBKMT2APPARG
SCHEMBL1892153 0.70 PPARG (0.46) MAPK14PPARG
SCHEMBL1894638 0.69 PPARG (0.56) PPARG
SCHEMBL4011554 0.69 PPARG (0.46) ALDH1A1MAPK14POLBKMT2APPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed