SCHEMBL4017239

SCHEMBL4017239

NCCCSC[C@H](N)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ARG1 P05089 1/20 0.58
ARG2 P78540 1/20 0.58
NOS2 P35228 3/20 0.57
GSR P00390 1/20 0.52
NOS1 P29475 2/20 0.51
NOS3 P29474 1/20 0.51
BHMT Q93088 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017246 1.00 ARG1 (0.58) ARG1ARG2NOS2GSRNOS1
Aspartic Acid SCHEMBL7373778 0.88 NOS2 (0.48) ARG1ARG2NOS2GSRNOS1
SCHEMBL296784 0.87 ARG1 (0.62) ARG1ARG2NOS2GSRNOS1
SCHEMBL9821119 0.87 ARG1 (0.62) ARG1ARG2NOS2GSRNOS1
SCHEMBL110108 0.87 ARG1 (0.62) ARG1ARG2NOS2GSRNOS1
Bromide SCHEMBL5505430 0.85 ARG1 (0.60) ARG1ARG2NOS2GSRNOS1
Bromide SCHEMBL5505432 0.85 ARG1 (0.60) ARG1ARG2NOS2GSRNOS1
Hydrochloric Acid SCHEMBL17633808 0.85 ARG1 (0.60) ARG1ARG2NOS2GSRNOS1
Hydrochloric Acid SCHEMBL9815370 0.85 ARG1 (0.60) ARG1ARG2NOS2GSRNOS1
Hydrochloric Acid SCHEMBL8472319 0.85 ARG1 (0.60) ARG1ARG2NOS2GSRNOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 149 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665853-B1 MULTIMERIC POLYVALENT ANTITHROMBOTIC AGENTS DIATIDE INC (US) 2002-08-14 EP claimed
EP-0693941-B1 RADIOLABELED COMPOUNDS FOR THROMBUS IMAGING DIATIDE INC (US) 2002-07-24 EP claimed
CN-1087630-C Radiolabeled compounds for imaging thrombi DIATECH INC (US) 2002-07-17 CN claimed
US-6136782-A LINEAR AND CYCLIC PEPTIDES THAT SPECIFICALLY BIND TO PLATELETS AND INHIBIT THEIR AGGREGATION DIATIDE, INC. (US) 2000-10-24 US claimed
US-6056940-A TECHNETIUM-99M COMPLEXING MOIETY COVALENTLY LINKED TO A PLATELET GLYCOPROTEIN IIB/IIIA RECEPTOR BINDING MOIETY HAVING A MOLECULAR WEIGHT OF LESS THAN 10,000 DALTONS DIATIDE, INC. (US) 2000-05-02 US claimed
US-5977064-A CYCLIC TETRAPEPTIDE AS ANTICOAGULANT DIATIDE, INC. (US) 1999-11-02 US claimed
US-5830856-A RADIOLABELED SCINTIGRAPHIC IMAGING DIATIDE, INC. (US) 1998-11-03 US claimed
CN-1154071-A Radiolabeled compounds for imaging thrombi DIATECH INC (US) 1997-07-09 CN claimed
EP-0665853-A1 MULTIMERIC POLYVALENT ANTITHROMBOTIC AGENTS Diatide, Inc. (US) 1995-08-09 EP claimed
WO-1994023758-A1 RADIOLABELED COMPOUNDS FOR THROMBUS IMAGING DIATECH, INC. (US) 1994-10-27 WO claimed
WO-1994007918-A1 MULTIMERIC POLYVALENT ANTITHROMBOTIC AGENTS DIATECH, INC. (US) 1994-04-14 WO claimed
EP-4531925-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF NEUROLOGICAL DISORDERS D&D Pharmatech Inc. (KR) 2025-04-09 EP disclosed
EP-4532530-A1 PEPTIDE COMPOSITIONS AND METHODS OF USE THREOF D&D Pharmatech Inc. (KR) 2025-04-09 EP disclosed
WO-2023228156-A1 PEPTIDE COMPOSITIONS AND METHODS OF USE THREOF D&D PHARMATECH INC. (KR) 2023-11-30 WO disclosed
WO-2023228155-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF NEUROLOGICAL DISORDERS D&D PHARMATECH INC. (KR) 2023-11-30 WO disclosed
WO-1994007918-A1 MULTIMERIC POLYVALENT ANTITHROMBOTIC AGENTS DIATECH, INC. (US) 1994-04-14 WO disclosed
WO-1994000489-A2 RADIOACTIVELY-LABELED SOMATOSTANTIN-DERIVED PEPTIDES FOR IMAGING AND THERAPEUTIC USES DIATECH, INC. (US) 1994-01-06 WO disclosed
WO-1993025244-A1 TECHNETIUM-99m LABELED PEPTIDES FOR IMAGING DIATECH, INC. (US) 1993-12-23 WO disclosed
WO-1993023085-A1 TECHNETIUM-99m LABELED PEPTIDES FOR THROMBUS IMAGING DIATECH, INC. (US) 1993-11-25 WO disclosed
WO-1993021962-A1 TECHNETIUM-99m LABELED PEPTIDES FOR IMAGING DIATECH, INC. (US) 1993-11-11 WO disclosed