SCHEMBL4017261

SCHEMBL4017261

CS(=O)(=O)c1cccc(-c2ccc(F)c(-c3ccnc4c(S(C)(=O)=O)cccc34)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 11/20 0.58
NR1H3 Q13133 11/20 0.58
RXRA P19793 1/20 0.48
CYP2C9 P11712 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.42
GLO1 Q04760 1/20 0.40
PLK4 O00444 2/20 0.40
SYK P43405 1/20 0.40
LIMK1 P53667 1/20 0.39
EPHB4 P54760 1/20 0.39
CCNT1 O60563 1/20 0.39
CDK9 P50750 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018063 0.87 NR1H2 (0.55) NR1H2NR1H3RXRACYP2C9PTGDR2
SCHEMBL4009593 0.86 NR1H2 (0.55) NR1H2NR1H3RXRASYKCCNT1
SCHEMBL4012639 0.86 NR1H2 (0.72) NR1H2NR1H3RXRACYP2C9PTGDR2
SCHEMBL4011973 0.84 NR1H2 (0.58) NR1H2NR1H3RXRAPTGDR2
SCHEMBL4299566 0.81 NR1H2 (0.50) NR1H2NR1H3RXRAPTGDR2GLO1
SCHEMBL4011406 0.81 CYP4F2 (0.44) NR1H2NR1H3RXRAPTGDR2CCNT1
SCHEMBL4017722 0.80 NR1H2 (0.74) NR1H2NR1H3RXRACYP2C9GLO1
SCHEMBL4010255 0.80 NR1H2 (0.48) NR1H2NR1H3RXRAPTGDR2GLO1
SCHEMBL27765021 0.77 NR1H2 (0.51) NR1H2NR1H3RXRAPTGDR2GLO1
SCHEMBL4010387 0.77 NR1H2 (0.48) NR1H2NR1H3RXRAPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed