SCHEMBL4299566

SCHEMBL4299566

CS(=O)(=O)c1cccc2c(-c3cc(O)ccc3F)ccnc12

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.50
NR1H3 Q13133 5/20 0.50
PTGDR2 Q9Y5Y4 1/20 0.47
COMT P21964 6/20 0.40
PIK3CD O00329 1/20 0.40
KDM4E B2RXH2 2/20 0.39
GLO1 Q04760 1/20 0.38
RXRA P19793 1/20 0.38
CCNT1 O60563 2/20 0.37
CDK9 P50750 2/20 0.37
ALPL P05186 1/20 0.36
ALPI P09923 1/20 0.36
ALPG P10696 1/20 0.36
DNMT1 P26358 1/20 0.36
MCL1 Q07820 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TOP2A P11388 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012181 0.85 PTGDR2 (0.45) NR1H2NR1H3PTGDR2COMTPIK3CD
SCHEMBL4010255 0.83 NR1H2 (0.48) NR1H2NR1H3PTGDR2GLO1RXRA
SCHEMBL4017261 0.81 NR1H2 (0.58) NR1H2NR1H3PTGDR2GLO1RXRA
SCHEMBL4018184 0.81 PIK3CD (0.54) NR1H2NR1H3PTGDR2PIK3CDGLO1
SCHEMBL17044085 0.80 KDR (0.46) NR1H2NR1H3PTGDR2COMTKDM4E
SCHEMBL4016970 0.80 NR1H3 (0.50) NR1H2NR1H3PTGDR2GLO1RXRA
SCHEMBL4011973 0.79 NR1H2 (0.58) NR1H2NR1H3PTGDR2RXRA
SCHEMBL4010284 0.79 NR1H2 (0.53) NR1H2NR1H3PTGDR2PIK3CDKDM4E
SCHEMBL4011406 0.78 CYP4F2 (0.44) NR1H2NR1H3PTGDR2RXRACCNT1
SCHEMBL17044115 0.78 KDM4E (0.44) NR1H2NR1H3PTGDR2COMTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed