SCHEMBL4018339

SCHEMBL4018339

S=c1nc(Cc2cccnc2)[nH][nH]1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
MMP2 P08253 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CACNA1H O95180 1/20 0.41
CHRNA7 P36544 1/20 0.41
CTSL P07711 1/20 0.41
TBXAS1 P24557 1/20 0.40
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
MPO P05164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8007687 0.73 MMP2 (0.47) HRH4HRH3MMP2ALDH1A1KDM4E
SCHEMBL727185 0.73 CYP1A2 (0.62) HRH4HRH3MMP2CYP1A2CYP2D6
SCHEMBL31688985 0.69 TAAR1 (0.68) HRH4HRH3MMP2CYP1A2CYP2D6
SCHEMBL6168636 0.69 TAAR1 (0.68) HRH4HRH3MMP2CYP1A2CYP2D6
SCHEMBL7370545 0.68 CYP2C19 (0.56) HRH4HRH3MMP2CYP1A2CYP2D6
SCHEMBL3335641 0.68 GAA (0.71) KDM4EGAACACNA1H
SCHEMBL29995759 0.68 CYP11B1 (0.65) HRH4HRH3CYP1A2CYP2D6CHRNA7
SCHEMBL177863 0.68 CYP11B1 (0.65) HRH4HRH3CYP1A2CYP2D6CHRNA7
SCHEMBL14257669 0.68 CYP1A2 (0.56) HRH4HRH3MMP2CYP1A2CYP2D6
SCHEMBL4016895 0.67 DCUN1D1 (0.63) ALDH1A1KDM4EGAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009087218-A1 THIAZOLTRIAZOLES AND THIAZOLIMIDAZOLES AS ANTAGONISTS OF THE MGLUR5 RECEPTOR GLAXO GROUP LIMITED (GB) 2009-07-16 WO disclosed