SCHEMBL8007687

SCHEMBL8007687

S=c1[nH]nc(Cc2cccnc2)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.47
HRH4 Q9H3N8 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
DAO P14920 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CACNA1H O95180 1/20 0.41
CYP2C19 P33261 1/20 0.41
CHRNA7 P36544 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
TBXAS1 P24557 1/20 0.40
LTA4H P09960 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28761060 0.80 DAO (0.62) ALDH1A1KDM4ESMN1; SMN2DAOCYP2C9
SCHEMBL4018339 0.73 HRH4 (0.46) MMP2HRH4HRH3ALDH1A1KDM4E
SCHEMBL727185 0.73 CYP1A2 (0.62) MMP2HRH4HRH3CYP1A2CYP2D6
SCHEMBL7370545 0.71 CYP2C19 (0.56) MMP2HRH4HRH3CYP1A2CYP2D6
SCHEMBL11427746 0.70 ALDH1A1 (0.50) HRH4HRH3ALDH1A1KDM4EHPGD
SCHEMBL6168636 0.69 TAAR1 (0.68) MMP2HRH4HRH3CYP1A2CYP2D6
SCHEMBL31688985 0.69 TAAR1 (0.68) MMP2HRH4HRH3CYP1A2CYP2D6
SCHEMBL14123294 0.69 SMN1; SMN2 (0.68) MMP2HRH4HRH3ALDH1A1SMN1; SMN2
SCHEMBL7007907 0.68 PNP (0.55) HRH4HRH3DAO
SCHEMBL23674843 0.68 MMP2 (0.45) MMP2HRH4HRH3ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009087218-A1 THIAZOLTRIAZOLES AND THIAZOLIMIDAZOLES AS ANTAGONISTS OF THE MGLUR5 RECEPTOR GLAXO GROUP LIMITED (GB) 2009-07-16 WO disclosed