SCHEMBL4018461

SCHEMBL4018461

COC(=O)C(F)(F)F.O=Cc1cccc2c1ccn2S(=O)(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 13/20 0.49
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
RORC P51449 1/20 0.41
BCHE P06276 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 1/20 0.39
UBE2N P61088 1/20 0.39
PPARG P37231 1/20 0.38
PPARD Q03181 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4018464 0.89 HTR6 (0.49) HTR6HDAC3HDAC4HDAC1HDAC7
SCHEMBL3623386 0.89 HTR6 (0.51) HTR6HDAC3HDAC4HDAC1HDAC7
SCHEMBL3613851 0.79 HTR6 (0.48) HTR6HDAC3HDAC4HDAC1HDAC7
Trifluoroacetic Acid SCHEMBL4021249 0.76 HTR6 (0.61) HTR6
Trifluoroacetic Acid SCHEMBL4018381 0.74 HTR6 (0.48) HTR6RORC
SCHEMBL3621863 0.73 HTR6 (0.50) HTR6RORCPPARGPPARDPPARA
SCHEMBL3619113 0.73 HTR6 (0.46) HTR6RORCBCHEKDM4E
SCHEMBL743239 0.72 HTR6 (0.64) HTR6HDAC3HDAC4HDAC1HDAC7
SCHEMBL6174821 0.72 HTR6 (0.55) HTR6RORCBCHE
Trifluoroacetic Acid SCHEMBL3625968 0.72 HTR6 (0.53) HTR6HDAC1HDAC2HDAC6RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046741-A1 INDOLES AS 5-HT6 MODULATORS BIOVITRUM AB (publ) (SE) 2009-04-15 EP disclosed
WO-2008003703-A1 INDOLES AS 5-HT6 MODULATORS BIOVITRUM AB (PUBL) (SE) 2008-01-10 WO disclosed