SCHEMBL4020465

SCHEMBL4020465

O=C(O)C(C(=O)C1CCC(C(F)(F)F)CC1)c1nc2ccccc2s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.45
HPGD P15428 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP2C9 P11712 1/20 0.45
HIF1A Q16665 1/20 0.45
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.42
TP53 P04637 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.42
ALOX5 P09917 1/20 0.39
ALDH1A1 P00352 7/20 0.39
POLB P06746 3/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13746880 0.87 GAA (0.41) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL11697365 0.72 HPGD (0.60) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL9306307 0.71 HPGD (0.58) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL9306298 0.71 HPGD (0.58) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL11191161 0.70 HPGD (0.60) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL1371913 0.69 HPGD (0.56) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL4021493 0.69 KDM4E (0.38) HPGDCYP2C19CYP2C9SMN1; SMN2MAPT
SCHEMBL5536307 0.68 HPGD (0.66) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL9306300 0.68 HPGD (0.62) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL5159135 0.67 HPGD (0.60) HSD17B10HPGDCYP1A2CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed