Theobromine

Theobromine

SCHEMBL4021232

Cn1cnc2c1c(=O)[nH]c(=O)n2C.[KH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.96
PMP22 Q01453 2/20 0.96
MAPK1 P28482 2/20 0.96
ADORA2A P29274 4/20 0.62
PDE4A P27815 3/20 0.62
PDE4B Q07343 3/20 0.62
PDE4C Q08493 3/20 0.62
PDE4D Q08499 3/20 0.62
LMNA P02545 2/20 0.53
ALDH1A1 P00352 2/20 0.53
MAPT P10636 1/20 0.53
TSHR P16473 1/20 0.53
BLM P54132 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.52
POLB P06746 2/20 0.51
GDA Q9Y2T3 2/20 0.51
PIK3CD O00329 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
CNR1 P21554 1/20 0.51
ACHE P22303 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Theobromine SCHEMBL11599459 0.98 CYP3A4 (1.00) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL3184 0.98 CYP3A4 (1.00) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL1690622 0.98 CYP3A4 (1.00) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL29658415 0.96 CYP3A4 (0.96) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL6062232 0.96 CYP3A4 (0.96) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL606388 0.96 CYP3A4 (0.96) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL7926330 0.96 CYP3A4 (0.96) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL1291169 0.96 CYP3A4 (0.96) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL28252424 0.96 CYP3A4 (0.96) CYP3A4PMP22MAPK1ADORA2APDE4A
Theobromine SCHEMBL16093810 0.95 CYP3A4 (0.93) CYP3A4PMP22MAPK1ADORA2APDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130052280-A1 USE OF THEBROMINE FOR LOWERING CENTRAL BLOOD PRESSURE CONOPCO,INC., D/B/A UNILEVER 2013-02-28 US claimed
JP-55143985-A None JP disclosed
US-20130052280-A1 USE OF THEBROMINE FOR LOWERING CENTRAL BLOOD PRESSURE CONOPCO,INC., D/B/A UNILEVER 2013-02-28 US disclosed
WO-2009089677-A1 THEOBROMINE PRODUCTION PROCESS PERRIGO TRADING (SHANGHAI) CO., LTD. (CN) 2009-07-23 WO disclosed
JP-S55143985-A PREPARATION OF NOVEL XANTHINE DERIVATIVE KYOWA HAKKO KOGYO CO LTD 1980-11-10 JP disclosed
US-4060618-A Quaternary xanthinylalkyl nortropine DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DT) 1977-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130052280-A1 USE OF THEBROMINE FOR LOWERING CENTRAL BLOOD PRESSURE APOB, BHMT, HDLBP CYP3A4 1262/4885PMP22 563/4885MAPK1 643/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.