SCHEMBL4021713

SCHEMBL4021713

C[C@@H]1CN(c2ccc(Cl)cc2)CCN1C(Cl)C=O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.40
SLC6A9 P48067 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
GSK3B P49841 1/20 0.37
POLB P06746 2/20 0.36
HPGD P15428 2/20 0.36
DRD4 P21917 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
MAPT P10636 1/20 0.36
LMNA P02545 2/20 0.35
ALDH1A1 P00352 1/20 0.35
AKR1C3 P42330 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014671 1.00 NOTUM (0.40) NOTUMSLC6A9SMN1; SMN2KMT2AMEN1
SCHEMBL19003591 0.81 SLC6A9 (0.43) NOTUMSLC6A9SMN1; SMN2KMT2AMEN1
SCHEMBL17897288 0.81 SLC6A9 (0.43) NOTUMSLC6A9SMN1; SMN2KMT2AMEN1
SCHEMBL3817807 0.80 CCR1 (0.44) MAPTLMNAALDH1A1
SCHEMBL4013778 0.74 HTR3E (0.46) SMN1; SMN2KMT2AMEN1POLBHPGD
SCHEMBL15858055 0.72 ADRA2A (0.52) NOTUMCYP1A2CYP2D6GSK3BPOLB
SCHEMBL17897287 0.72 ADRA2A (0.52) NOTUMCYP1A2CYP2D6GSK3BPOLB
SCHEMBL6169684 0.72 CCR1 (0.46)
SCHEMBL6171097 0.72 CCR1 (0.46)
SCHEMBL18948533 0.69 KMT2A (0.49) NOTUMSLC6A9KMT2AMEN1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1691810-A4 SUBSTITUTED PIPERAZINES CHEMOCENTRYX INC (US) 2009-07-01 EP disclosed
EP-1691810-A1 SUBSTITUTED PIPERAZINES ChemoCentryx Inc (US) 2006-08-23 EP disclosed
WO-2005056015-A1 SUBSTITUTED PIPERAZINES CHEMOCENTRYX, INC. (US) 2005-06-23 WO disclosed