SCHEMBL4023870

SCHEMBL4023870

CCC(=O)N(C)c1ccc(F)cn1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.39
HDAC1 Q13547 4/20 0.37
GRIN2B Q13224 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
POLB P06746 1/20 0.35
APEX1 P27695 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CXCR1 P25024 2/20 0.34
CXCR2 P25025 2/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
TDO2 P48775 1/20 0.34
PTGIR P43119 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15173773 0.81 HCAR3 (0.38) HCAR3HDAC1PTGDR2CXCR1CXCR2
SCHEMBL2790729 0.80 HCAR3 (0.39) HCAR3HDAC1TDP1ALDH1A1SYK
SCHEMBL4172587 0.73 HCAR3 (0.40) HCAR3HDAC1PTGDR2POLBGRIN1
SCHEMBL3718183 0.73 HDAC1 (0.37) HCAR3HDAC1GRIN1GRIN2APTGIR
SCHEMBL4782065 0.73 HDAC1 (0.37) HCAR3HDAC1GRIN2BCXCR1CXCR2
SCHEMBL13041524 0.73 POLQ (0.49) POLBAPEX1TDP1KDM4E
SCHEMBL15551126 0.72 POLQ (0.51) POLBKMT2A
SCHEMBL26508794 0.72 TDO2 (0.49) TDO2
SCHEMBL25436833 0.70 JAK2 (0.34) KMT2A
SCHEMBL14547837 0.69 TDO2 (0.36) HDAC1PTGDR2TDO2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095712-A2 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2009-08-06 WO disclosed