SCHEMBL4024702

SCHEMBL4024702

CCCn1c(=O)c(C(=O)OCC)cc2c(-c3ccc(Cl)cc3)n(-c3ccccc3Cl)nc21

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.48
PDE4B Q07343 2/20 0.45
TP53 P04637 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
CASP1 P29466 3/20 0.44
CASP7 P55210 3/20 0.44
PDE4A P27815 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 3/20 0.42
GAA P10253 2/20 0.42
HSD17B10 Q99714 2/20 0.42
GLA P06280 1/20 0.42
MAPK1 P28482 1/20 0.42
POLB P06746 1/20 0.42
CNR2 P34972 1/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4181240 0.92 CNR1 (0.49) CNR1PDE4BTP53RXFP1CASP1
SCHEMBL4020761 0.91 CNR1 (0.45) CNR1PDE4BTP53RXFP1CASP1
SCHEMBL4020673 0.90 CNR1 (0.52) CNR1CNR2
SCHEMBL4021209 0.85 CNR1 (0.47) CNR1CNR2
SCHEMBL4027019 0.84 CNR1 (0.46) CNR1CNR2
SCHEMBL4192532 0.84 CNR1 (0.46) CNR1CNR2
SCHEMBL4024237 0.84 KDM4E (0.48) CNR1ALDH1A1KDM4EHPGDMAPK1
SCHEMBL4017677 0.83 CNR1 (0.44) CNR1RXFP1CASP1CASP7ALDH1A1
SCHEMBL4020767 0.82 CNR1 (0.45) CNR1CNR2
SCHEMBL4027308 0.81 CNR1 (0.45) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095752-A1 FUSED PYRAZOLE DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-08-06 WO disclosed