SCHEMBL4026944

SCHEMBL4026944

CNc1cc(-c2cccc(F)c2)nc2ccc(-c3ccccc3Cl)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 2/20 0.47
NT5E P21589 2/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
MAP4K4 O95819 1/20 0.42
ACP1 P24666 5/20 0.41
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
PTGS2 P35354 1/20 0.39
BACE1 P56817 1/20 0.39
DHODH Q02127 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MAPK1 P28482 2/20 0.38
GABBR2 O75899 1/20 0.38
GABBR1 Q9UBS5 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028870 0.87 CYP1A2 (0.47) CLK4NT5EABCG2MAP4K4ACP1
SCHEMBL4031373 0.87 ABCG2 (0.52) NT5EABCG2MAP4K4ACP1DHODH
SCHEMBL4023370 0.85 NT5E (0.49) NT5EABCG2MAP4K4ACP1AURKA
SCHEMBL4026246 0.84 LMNA (0.50) CLK4NT5EABCG2MAP4K4ACP1
SCHEMBL4025241 0.84 ACP1 (0.44) NT5EABCG2MAP4K4ACP1DHODH
SCHEMBL4021555 0.84 NT5E (0.48) CLK4NT5EABCG2MAP4K4ACP1
SCHEMBL4025363 0.83 ABCG2 (0.48) NT5EABCG2MAP4K4ACP1DHODH
SCHEMBL4024602 0.82 PDE10A (0.50) CYP2C9
SCHEMBL4032492 0.80 NT5E (0.45) CLK4NT5EABCG2MAP4K4ACP1
SCHEMBL4816411 0.79 ABCG2 (0.52) NT5EABCG2MAP4K4ACP1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP disclosed