SCHEMBL4032492

SCHEMBL4032492

CNc1cc(-c2cccc(F)c2)nc2ccc(-c3cc(C)cc(Cl)c3)cc12

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.45
ABCG2 Q9UNQ0 1/20 0.41
MAP4K4 O95819 4/20 0.41
ACP1 P24666 4/20 0.38
CLK4 Q9HAZ1 2/20 0.38
DHODH Q02127 3/20 0.37
MAOB P27338 1/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4021555 0.93 NT5E (0.48) NT5EABCG2MAP4K4ACP1CLK4
SCHEMBL4023370 0.88 NT5E (0.49) NT5EABCG2MAP4K4ACP1DHODH
SCHEMBL4031373 0.85 ABCG2 (0.52) NT5EABCG2MAP4K4ACP1DHODH
SCHEMBL4025363 0.84 ABCG2 (0.48) NT5EABCG2MAP4K4ACP1DHODH
SCHEMBL4026944 0.80 CLK4 (0.47) NT5EABCG2MAP4K4ACP1CLK4
SCHEMBL4028870 0.79 CYP1A2 (0.47) NT5EABCG2MAP4K4ACP1CLK4
SCHEMBL4816411 0.78 ABCG2 (0.52) NT5EABCG2MAP4K4ACP1DHODH
SCHEMBL4823113 0.77 ABCG2 (0.48) ABCG2MAP4K4ACP1MAOBKDM4E
SCHEMBL4028750 0.77 ABCG2 (0.48) ABCG2MAP4K4ACP1MAOBKDM4E
SCHEMBL4029317 0.76 CLK4 (0.48) CLK4DHODHKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP disclosed