SCHEMBL4031373

SCHEMBL4031373

CNc1cc(-c2cccc(F)c2)nc2ccc(-c3ccccc3)cc12

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.52
MAP4K4 O95819 2/20 0.48
TRIM58 Q8NG06 1/20 0.48
NT5E P21589 2/20 0.47
DHODH Q02127 2/20 0.47
ACP1 P24666 5/20 0.46
MAOB P27338 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ADORA2A P29274 1/20 0.41
ACHE P22303 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4025363 0.96 ABCG2 (0.48) ABCG2MAP4K4TRIM58NT5EDHODH
SCHEMBL4023370 0.92 NT5E (0.49) ABCG2MAP4K4TRIM58NT5EDHODH
SCHEMBL4021555 0.89 NT5E (0.48) ABCG2MAP4K4TRIM58NT5EDHODH
SCHEMBL4028870 0.88 CYP1A2 (0.47) ABCG2MAP4K4NT5EDHODHACP1
SCHEMBL4026944 0.87 CLK4 (0.47) ABCG2MAP4K4NT5EDHODHACP1
SCHEMBL4816411 0.86 ABCG2 (0.52) ABCG2MAP4K4NT5EDHODHACP1
SCHEMBL4028750 0.85 ABCG2 (0.48) ABCG2MAP4K4ACP1MAOBMEN1
SCHEMBL4823113 0.85 ABCG2 (0.48) ABCG2MAP4K4ACP1MAOBMEN1
SCHEMBL4032492 0.85 NT5E (0.45) ABCG2MAP4K4NT5EDHODHACP1
SCHEMBL4029317 0.85 CLK4 (0.48) DHODHADORA1MEN1KMT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP disclosed