SCHEMBL4028250

SCHEMBL4028250

CC(C)(C)C(Cc1cc(-c2cccnc2F)c(S(=O)(=O)c2cccc(C=O)c2)s1)NC(=O)O

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 8/20 0.32
NAT1 P18440 1/20 0.32
GRM4 Q14833 1/20 0.31
CYP3A4 P08684 1/20 0.30
LIPG Q9Y5X9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654949 0.88 AGTR2 (0.33) AGTR2CYP3A4LIPG
SCHEMBL3806158 0.87 AGTR2 (0.32) AGTR2GRM4CYP3A4LIPG
Hydrochloric Acid SCHEMBL3645134 0.85 NAMPT (0.33) AGTR2LIPG
SCHEMBL3652361 0.85 AGTR2 (0.33) AGTR2CYP3A4LIPG
Hydrochloric Acid SCHEMBL3653186 0.83 AGTR2 (0.32) AGTR2
SCHEMBL3649952 0.83 ABCC9 (0.36) AGTR2LIPG
SCHEMBL3803071 0.83 KDM4E (0.33) AGTR2
SCHEMBL3804718 0.82 ABCC9 (0.36) AGTR2CYP3A4LIPG
SCHEMBL4120137 0.82 LIPG (0.32) NAT1GRM4LIPG
SCHEMBL3650556 0.81 NAMPT (0.35) AGTR2GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed