SCHEMBL4028394

SCHEMBL4028394

Cc1nc(C2CCC(C(F)(F)F)CC2)c(-c2ccc3sccc3c2)c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
SPR P35270 9/20 0.35
MDM2 Q00987 2/20 0.33
DYRK1A Q13627 1/20 0.33
GRIA1 P42261 1/20 0.33
CA12 O43570 2/20 0.32
ENPP1 P22413 1/20 0.32
PDE2A O00408 3/20 0.32
CA2 P00918 1/20 0.32
CYP17A1 P05093 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028389 1.00 BRD4 (0.38) BRD4CREBBPSPRMDM2DYRK1A
SCHEMBL13746821 0.87 BRD4 (0.36) BRD4CREBBPSPRDYRK1AGRIA1
SCHEMBL13747129 0.80 TYMS (0.38) CA12PDE2ACA2
SCHEMBL13746898 0.77 HSD11B1 (0.39) PDE2A
SCHEMBL13746091 0.77 DYRK1A (0.35) SPRDYRK1AGRIA1PDE2A
SCHEMBL4020404 0.76 PDE2A (0.49) GRIA1PDE2A
SCHEMBL13746667 0.76 PDE2A (0.37) SPRPDE2A
SCHEMBL4023129 0.75 PDE2A (0.37) SPRPDE2A
SCHEMBL4023133 0.75 PDE2A (0.37) SPRPDE2A
SCHEMBL13746127 0.75 IRAK4 (0.44) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed