SCHEMBL4020404

SCHEMBL4020404

Cc1nc([C@H]2CC[C@@H](C(F)(F)F)CC2)c(-c2ccc(C(F)(F)F)nc2)c(=O)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 9/20 0.49
MCHR1 Q99705 1/20 0.39
GRIA1 P42261 3/20 0.37
KDM5B Q9UGL1 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
PLAT P00750 1/20 0.34
PDE9A O76083 2/20 0.33
PIK3CA P42336 1/20 0.33
KCNH2 Q12809 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3R1 P27986 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13746667 0.87 PDE2A (0.37) PDE2API4KBPIK3CA
SCHEMBL13746012 0.85 PIK3CA (0.36) PDE2AKDM5BPI4KBPDE9APIK3CA
SCHEMBL4023133 0.84 PDE2A (0.37) PDE2API4KB
SCHEMBL4023129 0.84 PDE2A (0.37) PDE2API4KB
SCHEMBL13747129 0.82 TYMS (0.38) PDE2APLAT
SCHEMBL13746898 0.80 HSD11B1 (0.39) PDE2APDE9A
SCHEMBL13746627 0.78 USP1 (0.34) PDE2APIK3CA
SCHEMBL13746091 0.77 DYRK1A (0.35) PDE2AGRIA1
SCHEMBL4028389 0.76 BRD4 (0.38) PDE2AGRIA1
SCHEMBL4028394 0.76 BRD4 (0.38) PDE2AGRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed