SCHEMBL4029367

SCHEMBL4029367

CCCOc1ccc(I)cc1C(=O)NCCC(O)c1c[nH]c2ccc(F)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 1/20 0.37
NOTUM Q6P988 2/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
CNR2 P34972 1/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTR1A P08908 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HIF1A Q16665 1/20 0.37
SPR P35270 1/20 0.36
PYGL P06737 1/20 0.36
SLC6A4 P31645 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
MPO P05164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035244 0.85 SCN8A (0.39) SCN8ASCN10ANOTUMMTNR1AMTNR1B
SCHEMBL3935484 0.77 HTR2A (0.41) SCN8ASCN10ANOTUMMTNR1AMTNR1B
SCHEMBL4029370 0.76 HTR1A (0.42) SCN8ASCN10ANOTUMMTNR1AMTNR1B
SCHEMBL5149356 0.74 KDM4E (0.38) KDM4ECNR2MEN1KMT2A
SCHEMBL5149347 0.74 KDM4E (0.38) KDM4ECNR2MEN1KMT2A
SCHEMBL17242338 0.71 KCNH2 (0.48) SLC6A4MPO
SCHEMBL4035537 0.71 SCN8A (0.37) SCN8ASCN10ANOTUMMTNR1AMTNR1B
SCHEMBL4031716 0.70 SCN8A (0.36) SCN8ASCN10ANOTUMMTNR1AMTNR1B
SCHEMBL4034238 0.69 SCN8A (0.34) SCN8ASCN10AKDM4ENOTUMMTNR1A
SCHEMBL4033961 0.68 MPO (0.41) SCN8ASCN10AHTR1ASPRSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed