SCHEMBL4030895

SCHEMBL4030895

O=Cc1ccc(C=S)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.52
HSD17B10 Q99714 1/20 0.52
ALDH5A1 P51649 1/20 0.52
ABAT P80404 1/20 0.52
ALDH1A1 P00352 8/20 0.50
KDM4E B2RXH2 3/20 0.46
TYR P14679 1/20 0.46
CYP2A13 Q16696 1/20 0.46
ALDH1A3 P47895 2/20 0.42
ALDH3A1 P30838 1/20 0.42
EGFR P00533 1/20 0.41
TRIM24 O15164 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
MAPK1 P28482 1/20 0.40
PTGS2 P35354 1/20 0.40
RAB9A P51151 1/20 0.40
STS P08842 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4952649 0.83 ALDH1A1 (0.38) ALDH1A1
SCHEMBL4956384 0.83 CYP2A6 (0.69) CYP2A6HSD17B10ALDH5A1ABATALDH1A1
SCHEMBL31171 0.83 CYP2A6 (0.69) CYP2A6HSD17B10ALDH5A1ABATALDH1A1
Water SCHEMBL29197442 0.79 CYP2A6 (0.65) CYP2A6HSD17B10ALDH5A1ABATALDH1A1
Hydrochloric Acid SCHEMBL28807787 0.79 CYP2A6 (0.65) CYP2A6HSD17B10ALDH5A1ABATALDH1A1
Formaldehyde SCHEMBL20477527 0.76 CYP2A6 (0.61) CYP2A6HSD17B10ALDH5A1ABATALDH1A1
SCHEMBL1713358 0.75
SCHEMBL25288128 0.73 CYP2A6 (0.58) CYP2A6HSD17B10ALDH5A1ABATALDH1A1
SCHEMBL9004502 0.73 CYP2A6 (0.58) CYP2A6HSD17B10ALDH5A1ABATALDH1A1
SCHEMBL4195177 0.73 CYP2A6 (0.58) CYP2A6HSD17B10ALDH5A1ABATALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4631323-A DOPING WITH CHARGE TRANSFER COMPOUNDS HONEYWELL INC. (US) 1986-12-23 US claimed
EP-4157458-B1 TRIARYLPYRIDINE COMPOUNDS AND USE THEREOF FOR TREATING CANCER INST NAT SANTE RECH MED (FR) 2024-04-17 EP disclosed
CN-114716289-B Preparation method of chiral benzyl alcohol derivative 华中师范大学 2024-03-01 CN disclosed
US-20230212146-A1 TRIARYLPYRIDINE COMPOUNDS AND USE THEREOF FOR TREATING CANCER CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2023-07-06 US disclosed
CN-114716289-A Preparation method of chiral benzyl alcohol derivative 华中师范大学 2022-07-08 CN disclosed
CN-111937892-A Application of Aza-type isoalburnine derivative in prevention and treatment of agricultural plant diseases 兰州大学 2020-11-17 CN disclosed
CN-111233706-A Green synthesis method of sulindac 安徽峆一药业股份有限公司 2020-06-05 CN disclosed
EP-1363635-B1 SUBSTITUTED 8-ARYLQUINOLINE PHOSPHODIESTERASE-4 INHIBITORS MERCK & CO INC (US) 2009-04-15 EP disclosed
US-20090042888-A1 Prostaglandin endoperoxide H synthase biosynthesis inhibitors BLACK LAWRENCE A 2009-02-12 US disclosed
US-7427635-B2 Substituted hydantoins HOFFMANN-LA ROCHE INC. (US) 2008-09-23 US disclosed
US-5691373-A TREATING SUBARACHNOID HEMORRHAGE WARNER-LAMBERT COMPANY (US) 1997-11-25 US disclosed
EP-0772601-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-05-14 EP disclosed
US-5620999-A ANTIARTHRITIC, ANALGESIC AND ANTIPYRATIC AGENT G.D. SEARLE & CO. 1997-04-15 US disclosed
EP-0714391-A1 SUBSTITUTED 2(5H)FURANONE, 2(5H)THIOPHENONE AND 2(5H)PYRROLONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ENDOTHELIN ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1996-06-05 EP disclosed
WO-1996003387-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed
EP-0624159-A4 PYRIDYL SUBSTITUTED IMIDAZOLES. SMITHKLINE BEECHAM CORP (US) 1995-04-12 EP disclosed
WO-1995005376-A1 SUBSTITUTED 2(5H)FURANONE, 2(5H)THIOPHENONE AND 2(5H)PYRROLONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ENDOTHELIN ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1995-02-23 WO disclosed
EP-0624159-A1 PYRIDYL SUBSTITUTED IMIDAZOLES SMITHKLINE BEECHAM CORPORATION (US) 1994-11-17 EP disclosed
WO-1993014082-A1 PYRIDYL SUBSTITUTED IMIDAZOLES SMITHKLINE BEECHAM CORPORATION (US) 1993-07-22 WO disclosed
EP-0433662-A2 Acat inhibitors WARNER-LAMBERT COMPANY (US) 1991-06-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090042888-A1 Prostaglandin endoperoxide H synthase biosynthesis inhibitors PTGIS, PTGS1, PTGS2 CYP2A6 90/4885HSD17B10 234/4885ALDH5A1 95/4885
US-20230212146-A1 TRIARYLPYRIDINE COMPOUNDS AND USE THEREOF FOR TREATING CANCER TPX2, BRD4, BET1 CYP2A6 2948/4885HSD17B10 4789/4885ALDH5A1 3232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.