SCHEMBL4030980

SCHEMBL4030980

Cc1noc(-c2ccc(OC(F)(F)F)cc2)c1N(C(=O)O)C(C)c1ccccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38
SERPINE1 P05121 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
LPAR1 Q92633 2/20 0.34
LPAR3 Q9UBY5 2/20 0.34
LIPE Q05469 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
TRPM8 Q7Z2W7 3/20 0.34
PPARD Q03181 2/20 0.33
PPARA Q07869 2/20 0.33
P2RY2 P41231 1/20 0.33
P2RY1 P47900 1/20 0.33
P2RY14 Q15391 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030024 0.90 LPAR1 (0.42) IP6K1IP6K3IP6K2SERPINE1TRPV1
SCHEMBL4034800 0.90 TRPV1 (0.38) IP6K1IP6K3IP6K2SERPINE1TRPV1
SCHEMBL4030691 0.88 LPAR1 (0.41) IP6K1IP6K3IP6K2SERPINE1TRPV1
SCHEMBL4034111 0.87 BRD4 (0.37) IP6K1IP6K3IP6K2NPSR1TP53
SCHEMBL4033264 0.83 LPAR1 (0.40) NPSR1TP53MAPTLPAR1LPAR3
SCHEMBL4029114 0.81 HDAC6 (0.40) NPSR1TP53MAPTLPAR1LPAR3
SCHEMBL4034287 0.80 SLC16A3 (0.37) IP6K1IP6K3IP6K2LPAR1LPAR3
SCHEMBL4033894 0.78 LPAR1 (0.44) NPSR1MAPTLPAR1LPAR3GPBAR1
SCHEMBL4032476 0.77 LPAR1 (0.43) MAPTLPAR1LPAR3GPBAR1LPAR2
SCHEMBL4030221 0.77 LPAR1 (0.58) IP6K1IP6K3IP6K2TRPV1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed