SCHEMBL4031484

SCHEMBL4031484

COc1cccc(ON(C(=O)OC(C)(C)C)C(I)Cc2cccc(C(=O)N3CCN(C(C)C)CC3)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
ALDH1A1 P00352 9/20 0.42
PKM P14618 1/20 0.42
KDM4E B2RXH2 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13503924 0.75 ALDH1A1 (0.69) SLC6A2SLC6A4SLC6A3HRH3KMT2A
SCHEMBL4013523 0.74 HRH3 (0.68) SLC6A2SLC6A4SLC6A3HRH3ALDH1A1
SCHEMBL20812317 0.72 ACACB (0.54) SLC6A2SLC6A4SLC6A3HRH3KMT2A
SCHEMBL4374335 0.70 HRH3 (0.33) SLC6A2SLC6A4SLC6A3HRH3NPSR1
SCHEMBL20805385 0.70 HRH3 (0.52) SLC6A2SLC6A4SLC6A3HRH3KMT2A
SCHEMBL19605006 0.69 HRH3 (0.59) HRH3KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL19464759 0.69 ALDH1A1 (0.57) SLC6A2SLC6A4SLC6A3HRH3KMT2A
SCHEMBL23102110 0.68 HRH3 (0.55) HRH3KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL28759342 0.65 CRBN (0.53) KMT2AMEN1ALDH1A1PKMKDM4E
SCHEMBL13503762 0.65 EPHX2 (0.61) HRH3KMT2AMEN1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049473-A2 SUBSTITUTED BENZYL AMINE COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2009-04-22 EP disclosed
WO-2008002820-A2 SUBSTITUTED BENZYL AMINE COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2008-01-03 WO disclosed